Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily M member 8' and Ligand = 'BDBM50241315'
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50241315((Z)-3-butylideneisobenzofuran-1(3H)-one | CHEMBL24...)
Affinity DataIC50:  1.41E+5nMAssay Description:Antagonist activity at rat recombinant TRPM8 overexpressed in HEK293 cells assessed as inhibition of icilin-induced intracellular calcium influx prei...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50241315((Z)-3-butylideneisobenzofuran-1(3H)-one | CHEMBL24...)
Affinity DataIC50:  1.53E+5nMAssay Description:Antagonist activity at rat recombinant TRPM8 overexpressed in HEK293 cells assessed as inhibition of menthol-induced intracellular calcium influx pre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed