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Found 2 Enz. Inhib. hit(s) with Target = 'Transthyretin' and Ligand = 'BDBM576408'
TargetTransthyretin(Homo sapiens (Human))
Pfizer

WIPO
LigandPNGBDBM576408(4-(3,5-dimethyl- 1H-pyrazol-4-yl)-6-methyl-1,3-ben...)
Affinity DataKd:  58nMAssay Description:Affinity and Reversibility -The binding affinity and kinetics of binding were measured using Surface Plasmon Resonance based binding assay. These exp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTransthyretin(Homo sapiens (Human))
Pfizer

WIPO
LigandPNGBDBM576408(4-(3,5-dimethyl- 1H-pyrazol-4-yl)-6-methyl-1,3-ben...)
Affinity DataEC50:  21nMAssay Description:TTR SPA binding assays were performed in a final volume of 60 mI containing 100 ng human TTR (biotinylated recombinant protein) coupled to 25 pg SPA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed