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Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase BTK [C481S]' and Ligand = 'BDBM634113'
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Medshine Discovery

US Patent
LigandPNGBDBM634113(BDBM634121 | US20230357248, Example 4)
Affinity DataIC50:  7.30nMAssay Description:The specific assay process of BTK enzyme activity assay is as follows: Buffer: 20 mM 2-[4-(2-hydroxyethyl)-1-piperazinyl]ethanesulfonic acid (Hepes) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK [C481S](Homo sapiens (Human))
Medshine Discovery

US Patent
LigandPNGBDBM634113(BDBM634121 | US20230357248, Example 4)
Affinity DataIC50:  15.1nMAssay Description:The specific assay process of BTK enzyme activity assay is as follows: Buffer: 20 mM 2-[4-(2-hydroxyethyl)-1-piperazinyl]ethanesulfonic acid (Hepes) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent