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Report error Found 2 Enz. Inhib. hit(s) with Target = 'Ubiquitin carboxyl-terminal hydrolase 8' and Ligand = 'BDBM50597453'
TargetUbiquitin carboxyl-terminal hydrolase 8(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50597453(CHEMBL4567355)
Affinity DataIC50:  3.16E+4nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50597453(CHEMBL4567355)
Affinity DataKd:  4.36E+4nMAssay Description:Binding affinity to N-terminal His6-tagged USP8 catalytic domain (734 to 1110 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed