Found 2 Enz. Inhib. hit(s) with Target = 'Vitamin D3 receptor' and Ligand = 'BDBM50455855' TargetVitamin D3 receptor(Homo sapiens (Human))
University of Santiago De Compostela
Curated by ChEMBL
University of Santiago De Compostela
Curated by ChEMBL
Affinity DataIC50: 5.60nMAssay Description:Displacement of fluormone from human full length VDR after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
University of Santiago De Compostela
Curated by ChEMBL
University of Santiago De Compostela
Curated by ChEMBL
Affinity DataEC50: 8.60nMAssay Description:Agonist activity at VDR in human MCF7 cells assessed as increase in transcription of CYP24A1 gene after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
