Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'cAMP-dependent protein kinase catalytic subunit alpha' and Ligand = 'BDBM2706'
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
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LigandPNGBDBM2706(3-[7-(aminomethyl)-6H,7H,8H,9H,10H-azepino[1,2-a]i...)
Affinity DataIC50:  1.28E+4nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed