Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50014198
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50105329(CHEMBL1213492)
Affinity DataIC50:  70nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50573502(CHEMBL4870227)
Affinity DataIC50:  718nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50531020(CHEMBL4448410)
Affinity DataIC50:  924nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50531013(CHEMBL4453121)
Affinity DataIC50:  930nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50531057(CHEMBL4448978)
Affinity DataIC50:  1.91E+3nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50573498(CHEMBL4852256)
Affinity DataIC50:  3.06E+3nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50573501(CHEMBL4862508)
Affinity DataIC50:  3.21E+3nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50531051(CHEMBL4470373)
Affinity DataIC50:  3.96E+3nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50015181(CHEMBL154302 | N-Hydroxy-4-methyl-benzamide)
Affinity DataIC50:  5.64E+3nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50573495(CHEMBL4873055)
Affinity DataIC50:  6.83E+3nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50573491(CHEMBL4862563)
Affinity DataIC50:  7.09E+3nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50025840(4-Amino-N-hydroxy-benzamide | 4-aminobenzohydroxam...)
Affinity DataIC50:  7.14E+3nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50573499(CHEMBL4869421)
Affinity DataIC50:  7.39E+3nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50573497(CHEMBL4864065)
Affinity DataIC50:  9.71E+3nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50573494(CHEMBL4877419)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50573496(CHEMBL4863455)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50573500(CHEMBL4851389)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50015184(BENZHYDROXAMIC ACID | BENZOHYDROXAMATE | CHEMBL163...)
Affinity DataIC50:  2.54E+4nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50573493(CHEMBL4850382)
Affinity DataIC50:  2.94E+4nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Italfarmaco

Curated by ChEMBL
LigandPNGBDBM50573492(NSC-13997 | Nicoxamat)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of recombinant human C-terminal His-tagged HDAC1 expressed in Sf9 insect cells using Fluor de Lys deacetylase or Fluor de Lys Green deacet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed