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Report error Found 17 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50045745
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079375(CHEMBL3417008 | US9663465, 20)
Affinity DataKi:  0.950nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079377(CHEMBL3417007)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079367(CHEMBL3416998)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079365(CHEMBL3416996 | US9663465, 8)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079366(CHEMBL3416997 | US9663465, 12)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079369(CHEMBL3417000 | US9663465, 11)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079362(CHEMBL3417009 | US9663465, 9)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079368(CHEMBL3416999 | US9663465, 16)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079364(CHEMBL3416995 | US9663465, 7)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM84950(CAS_183782 | NSC_183782 | RS 67333)
Affinity DataKi:  9.30nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079370(CHEMBL3417001)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079363(CHEMBL3414597 | US9663465, 6)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079371(CHEMBL3417002)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079372(CHEMBL3417003)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079376(CHEMBL3417005)
Affinity DataKi:  105nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079374(CHEMBL3417006)
Affinity DataKi:  122nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Cermn

Curated by ChEMBL
LigandPNGBDBM50079373(CHEMBL3417004)
Affinity DataKi:  193nMAssay Description:Displacement of [3H]GR113808 from 5-HT4R in guinea pig brain membranes incubated for 30 mins by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed