Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with all data for assayid = 8 entry = 50009557
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50529882(CHEMBL1236255)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of recombinant human His6-tagged N-terminal PDHK2 (A8 to T399 residues) expressed in baculovirus expression system using PDC as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Jiangsu Normal University

Curated by ChEMBL
LigandPNGBDBM50529882(CHEMBL1236255)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of recombinant human His6-tagged N-terminal PDHK2 (A8 to T399 residues) expressed in baculovirus expression system using PDC as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB