Affinity DataKi: 19nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibition of human CYP2C9More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 65nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 81nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
Affinity DataKi: 410nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.02E+3nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.07E+3nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
Affinity DataKi: 2.77E+3nMAssay Description:Inhibition of human dopamine D3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.77E+3nMAssay Description:Inhibition of human dopamine D3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.77E+3nMAssay Description:Inhibition of human dopamine D3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.77E+3nMAssay Description:Inhibition of human dopamine D3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
Affinity DataKi: 4.50E+3nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
Affinity DataKi: 4.50E+3nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:Inhibition of human dopamine D2L receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.50E+3nMAssay Description:Inhibition of human dopamine D2L receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.20E+3nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
Affinity DataKi: 1.08E+4nMAssay Description:Inhibition of human dopamine D3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:Inhibition of human CYP2C19More data for this Ligand-Target Pair
Affinity DataKi: 1.57E+4nMAssay Description:Inhibition of human dopamine D3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.59E+4nMAssay Description:Inhibition of human dopamine D3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Northwest Agriculture & Forestry University
Curated by ChEMBL
Northwest Agriculture & Forestry University
Curated by ChEMBL
Affinity DataIC50: 66nMAssay Description:Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a...More data for this Ligand-Target Pair
TargetHigh affinity choline transporter 1(Homo sapiens (Human))
Vanderbilt University Medical Center
Curated by ChEMBL
Vanderbilt University Medical Center
Curated by ChEMBL
Affinity DataIC50: 72nMAssay Description:Inhibition of [3H]choline uptake at human choline transporter expressed in HEK293 cells preincubated for 15 mins followed by [3H]choline addition mea...More data for this Ligand-Target Pair
TargetHigh affinity choline transporter 1(Homo sapiens (Human))
Vanderbilt University Medical Center
Curated by ChEMBL
Vanderbilt University Medical Center
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of human CHT Leu530Ala and Val531Ala mutant expressed in HEK293 cells assessed as remaining transporter activity in presence of 10 uM [3H]...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
TargetHigh affinity choline transporter 1(Homo sapiens (Human))
Vanderbilt University Medical Center
Curated by ChEMBL
Vanderbilt University Medical Center
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human CHT Leu530Ala and Val531Ala mutant expressed in HEK293 cells assessed as remaining transporter activity in presence of 10 uM [3H]...More data for this Ligand-Target Pair