Compile Data Set for Download or QSAR
Report error Found 4 of ic50 for UniProtKB: P32297
LigandChemical structure of BindingDB Monomer ID 50445325BDBM50445325(CHEMBL3104238)
Affinity DataIC50: 0.950nMAssay Description:Antagonist activity at human alpha6/alpha3beta2beta3 nAChR expressed in Xenopus oocytes assessed as inhibition of ACh-induced current by voltage clam...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50170585BDBM50170585(CHEMBL406906)
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against Nicotinic acetylcholine receptor alpha-6-alpha-3-beta-2-beta-3; Range is 0.7-1 nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50567435BDBM50567435(CHEMBL4872191)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of human alpha6/alpha3beta2beta3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current respons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50567433BDBM50567433(CHEMBL4869892)
Affinity DataIC50: 135nMAssay Description:Inhibition of human alpha6/alpha3beta2beta3 nAChR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced current respons...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed