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Report error Found 132 of ki for UniProtKB: P48039
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118462BDBM50118462(2,2,2-Trifluoro-N-[2-(6-methoxy-2-phenyl-3H-inden-...)
Affinity DataKi:  0.00602nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118435BDBM50118435(2,2,2-Trifluoro-N-[2-(6-methoxy-indan-1-yl)-ethyl]...)
Affinity DataKi:  0.0123nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471134BDBM50471134(CHEMBL64664)
Affinity DataKi:  0.0140nMAssay Description:Displacement of 2-[125I]iodomelatonin from melatonin receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471125BDBM50471125(CHEMBL433237)
Affinity DataKi:  0.0140nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin (100 pM) as labelled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50034110BDBM50034110(Melatonin,2-Phenyl | CHEMBL15060 | N-[2-(5-Methoxy...)
Affinity DataKi:  0.0170nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin (100 pM) as labelled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50034110BDBM50034110(Melatonin,2-Phenyl | CHEMBL15060 | N-[2-(5-Methoxy...)
Affinity DataKi:  0.0170nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin as labelled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 29611BDBM29611(CHEMBL289233 | Melatonin,2-Iodo | 2-Iodomelatonin)
Affinity DataKi:  0.0210nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to melatonin receptor in quail brain as 1/KaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118446BDBM50118446(2,2,2-Trifluoro-N-[2-(6-methoxy-indan-1-yl)-ethyl]...)
Affinity DataKi:  0.0225nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118456BDBM50118456(N-[2-(6-Methoxy-3H-inden-1-yl)-ethyl]-propionamide...)
Affinity DataKi:  0.0231nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118453BDBM50118453((S) N-[2-(6-Methoxy-indan-1-yl)-ethyl]-butyramide ...)
Affinity DataKi:  0.0321nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50043287BDBM50043287(Melatonin,2-Bromo | N-[2-(2-Bromo-5-methoxy-1H-ind...)
Affinity DataKi:  0.0360nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin (100 pM) as labelled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50043287BDBM50043287(Melatonin,2-Bromo | N-[2-(2-Bromo-5-methoxy-1H-ind...)
Affinity DataKi:  0.0360nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin as labelled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118440BDBM50118440(2,2,2-Trifluoro-N-[2-(6-methoxy-3H-inden-1-yl)-eth...)
Affinity DataKi:  0.0408nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118430BDBM50118430((S) N-[2-(6-Methoxy-indan-1-yl)-ethyl]-propionamid...)
Affinity DataKi:  0.0410nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50506044BDBM50506044(CHEMBL4531537)
Affinity DataKi:  0.0440nMAssay Description:Displacement of 2-[125I]iodomelatonin from melatonin receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471136BDBM50471136(CHEMBL33006)
Affinity DataKi:  0.0440nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin (100 pM) as labelled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118463BDBM50118463(2,2,2-Trifluoro-N-[2-(7-methoxy-1,2,3,4-tetrahydro...)
Affinity DataKi:  0.0469nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118450BDBM50118450(N-[2-(6-Methoxy-indan-1-yl)-ethyl]-butyramide | CH...)
Affinity DataKi:  0.0553nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50034110BDBM50034110(Melatonin,2-Phenyl | CHEMBL15060 | N-[2-(5-Methoxy...)
Affinity DataKi:  0.0570nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to melatonin receptor in quail brain as 1/KaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50043287BDBM50043287(Melatonin,2-Bromo | N-[2-(2-Bromo-5-methoxy-1H-ind...)
Affinity DataKi:  0.0580nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to melatonin receptor in quail brain as 1/KaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118458BDBM50118458(N-[2-(6-Methoxy-indan-1-yl)-ethyl]-propionamide | ...)
Affinity DataKi:  0.0728nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118460BDBM50118460((S) N-[2-(6-Methoxy-indan-1-yl)-ethyl]-acetamide |...)
Affinity DataKi:  0.0733nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 9019BDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.0823nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 9019BDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.0915nMAssay Description:Binding affinity against ovine pars tuberalis melatonin receptor using 2-[125I]- melatonin radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2018
Entry Details

TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118436BDBM50118436(2,2,2-Trifluoro-N-[2-(6-methoxy-5-methyl-indan-1-y...)
Affinity DataKi:  0.0984nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50035179BDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataKi:  0.100nMAssay Description:Binding affinity against ovine pars tuberalis melatonin receptor using 2-[125I]- melatonin radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2018
Entry Details
PDB3D3D Structure (crystal)
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118447BDBM50118447(N-[2-(6-Ethoxy-indan-1-yl)-ethyl]-propionamide | C...)
Affinity DataKi:  0.100nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118441BDBM50118441(N-[2-(6-Methoxy-indan-1-yl)-ethyl]-acetamide | CHE...)
Affinity DataKi:  0.131nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50286970BDBM50286970(N-[2-(3H-Benzo[f]chromen-10-yl)-ethyl]-acetamide |...)
Affinity DataKi:  0.137nMAssay Description:Binding affinity against ovine pars tuberalis melatonin receptor using 2-[125I]- melatonin radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2018
Entry Details

TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 9019BDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.140nMAssay Description:Displacement of [125L]iodomelatonin from human MT1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471833BDBM50471833(CHEMBL127337)
Affinity DataKi:  0.176nMAssay Description:Binding affinity for Melatonin receptor using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118438BDBM50118438((E) N-[2-(6-Methoxy-indan-1-ylidene)-ethyl]-propio...)
Affinity DataKi:  0.208nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469786BDBM50469786(CHEMBL341392)
Affinity DataKi:  0.210nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to melatonin receptor in quail brain as 1/KaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50286973BDBM50286973(N-[2-(2,3-Dihydro-1H-benzo[f]chromen-10-yl)-ethyl]...)
Affinity DataKi:  0.216nMAssay Description:Binding affinity against ovine pars tuberalis melatonin receptor using 2-[125I]- melatonin radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2018
Entry Details

TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50506045BDBM50506045(CHEMBL4475742)
Affinity DataKi:  0.230nMAssay Description:Displacement of 2-[125I]iodomelatonin from melatonin receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471127BDBM50471127(CHEMBL62088)
Affinity DataKi:  0.230nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin (100 pM) as labelled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469784BDBM50469784(CHEMBL14975)
Affinity DataKi:  0.240nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to melatonin receptor in quail brain as 1/KaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118445BDBM50118445(N-[2-(6-Methoxy-indan-1-yl)-ethyl]-isobutyramide |...)
Affinity DataKi:  0.25nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471112BDBM50471112(CHEMBL61991)
Affinity DataKi:  0.390nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin as labelled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 9019BDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.410nMAssay Description:Displacement of [125L]iodomelatonin from human MT2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2016
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118452BDBM50118452(N-[2-(6-Propoxy-indan-1-yl)-ethyl]-propionamide | ...)
Affinity DataKi:  0.425nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469787BDBM50469787(CHEMBL127069)
Affinity DataKi:  0.430nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to melatonin receptor in quail brain as 1/KaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471119BDBM50471119(CHEMBL61380)
Affinity DataKi:  0.480nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin as labelled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118444BDBM50118444(2,2,2-Trifluoro-N-[3-(6-methoxy-indan-1-yl)-propyl...)
Affinity DataKi:  0.526nMAssay Description:Ability to inhibit 2-[125I]iodomelatonin specific binding to human melatonin receptor type 1A (MT1) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 9019BDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.610nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin as labelled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 9019BDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.610nMAssay Description:Displacement of 2-[125I]iodomelatonin from melatonin receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 9019BDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.610nMAssay Description:Binding affinity against melatonin receptor in the quail optica tecta using 2-[125] iodomelatonin (100 pM) as labelled ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 9019BDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.610nMAssay Description:Binding affinity for Melatonin receptor using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50469785BDBM50469785(CHEMBL130759)
Affinity DataKi:  0.630nMAssay Description:Inhibition of 2-[125I]iodomelatonin binding to melatonin receptor in quail brain as 1/KaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B(Human)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50286972BDBM50286972(N-(2-Naphtho[2,1-b]furan-9-yl-ethyl)-acetamide | C...)
Affinity DataKi:  0.780nMAssay Description:Binding affinity against ovine pars tuberalis melatonin receptor using 2-[125I]- melatonin radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2018
Entry Details

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