Compile Data Set for Download or QSAR
Report error Found 9 of ic50 for UniProtKB: P29274
TargetAdenosine receptor A2a/A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50182282(CHEMBL3818905)
Affinity DataIC50: 50nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2017
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50182281(CHEMBL3818205)
Affinity DataIC50: 70nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2017
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50182283(CHEMBL3819313)
Affinity DataIC50: 120nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2017
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50182284(CHEMBL3818888)
Affinity DataIC50: 250nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2017
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM81818(CHEMBL1909810 | NSC_1794 | CAS_1794 | HMA)
Affinity DataIC50: 270nMAssay Description:Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2017
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataIC50: 656nMAssay Description:Compound was evaluated for inhibition of adenosine induced relaxation against guinea-pig aorta (Adenosine A2 receptor).More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetAdenosine receptor A2a/A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50287703((E)-1-[(S)-2-(2-Hydroxy-ethyl)-piperidin-1-yl]-3-(...)
Affinity DataIC50: 1.18E+3nMAssay Description:Compound was evaluated for inhibition of adenosine induced relaxation against guinea-pig aorta (Adenosine A2 receptor).More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetAdenosine receptor A2a/A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50368346(CHEMBL608008)
Affinity DataIC50: 1.35E+4nMAssay Description:Maximal NECA stimulation of adenylate cyclase via Adenosine A2 receptor in human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a/A2b(Human)
Leiden University

Curated by ChEMBL
LigandPNGBDBM50079652((E)-1-[(R)-2-(2-Hydroxy-ethyl)-piperidin-1-yl]-3-(...)
Affinity DataIC50: 1.00E+5nMAssay Description:Compound was evaluated for inhibition of adenosine induced relaxation against guinea-pig aorta (Adenosine A2 receptor).More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article