Compile Data Set for Download or QSAR
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Found 3 of ec50 for monomerid = 21132
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University of Arizona Tucson

LigandPNGBDBM21132((3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-...)
Affinity DataKi:  1.60nM EC50:  4.60nMAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Arizona Tucson

LigandPNGBDBM21132((3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-...)
Affinity DataKi:  39nM ΔG°:  -42.3kJ/mole EC50:  18nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Arizona Tucson

LigandPNGBDBM21132((3S)-3-[(2S)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-...)
Affinity DataKi:  2.20nM ΔG°:  -49.4kJ/mole EC50:  120nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed