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Found 4 of ec50 for monomerid = 227552
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM227552(US9339486, CP55,940)
Affinity DataEC50:  0.140nMAssay Description:The compound of Example 3 was tested for agonist activity at the rat CB1 (rCB1) and rCB2 receptors, at eight concentrations, in duplicate: 10, 3, 1, ...More data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM227552(US9339486, CP55,940)
Affinity DataEC50:  1.13nMAssay Description:The compound of Example 3 was tested for agonist activity at the rat CB1 (rCB1) and rCB2 receptors, at eight concentrations, in duplicate: 10, 3, 1, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCannabinoid receptor 2(Homo sapiens (Human))
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM227552(US9339486, CP55,940)
Affinity DataEC50:  6.5nMAssay Description:Functional activity was evaluated using GTPγ[35S] assay in CHO membrane extracts expressing recombinant hCB1 (human CB1) receptors or hCB2 (huma...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
The Cleveland Clinic Foundation

US Patent
LigandPNGBDBM227552(US9339486, CP55,940)
Affinity DataEC50:  9nMAssay Description:Functional activity was evaluated using GTPγ[35S] assay in CHO membrane extracts expressing recombinant hCB1 (human CB1) receptors or hCB2 (huma...More data for this Ligand-Target Pair