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Found 3 of ec50 for monomerid = 292489
LigandPNGBDBM292489((S)-N-(2-(diethylamino)propyl)-2-(3-hydroxyazetidi...)
Affinity DataEC50:  6.20nMAssay Description:Inhibition of CaMK2gamma/delta in neonatal rat ventricular myocytes assessed as phospholamban phosphorylation after 4 hrs by Hoechst 33342 fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCalcium/calmodulin-dependent protein kinase type II subunit delta(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM292489((S)-N-(2-(diethylamino)propyl)-2-(3-hydroxyazetidi...)
Affinity DataEC50:  17.7nMAssay Description:CaMKII activity in neonatal rat ventricular myocytes (NRVM) was measured by monitoring the phosphorylation level of phospholamban using high-content ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
LigandPNGBDBM292489((S)-N-(2-(diethylamino)propyl)-2-(3-hydroxyazetidi...)
Affinity DataEC50:  274nMAssay Description:Inhibition of CaMK2alpha/beta in neonatal rat cortical neurons assessed as phospholamban phosphorylation after 4 hrs by Hoechst 33342 fluorescence-ba...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB