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Found 2 of ec50 for monomerid = 50105997
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105997(CHEMBL3598064)
Affinity DataEC50:  22nMAssay Description:Inverse agonist activity at RORgamma (unknown origin) transfected in HEK293T cells after 16 to 20 hrs by GAL4 luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-gamma(Mus musculus)
Biogen

Curated by ChEMBL
LigandPNGBDBM50105997(CHEMBL3598064)
Affinity DataEC50:  148nMAssay Description:Inverse agonist activity at RORgamma in C57BL/6 mouse splenocytes assessed as reduction of IL-17 production after 2 days by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed