Affinity DataEC50: 2nMAssay Description:Inverse agonist activity at RORgammat in mouse Th17 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Inverse agonist activity at RORgammat in CD3 and CD28-stimulated human whole blood assessed as reduction in IL17A production incubated for 1 hr befor...More data for this Ligand-Target Pair
Affinity DataEC50: >7.50E+3nMAssay Description:Inverse agonist activity of LXRbeta (unknown origin)More data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
Bristol Myers Squibb
Curated by ChEMBL
Bristol Myers Squibb
Curated by ChEMBL
Affinity DataEC50: 9.20E+3nMAssay Description:Inverse agonist activity of PXR (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of GAL4-fused RORalpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of GAL4-fused RORbeta (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: >1.20E+4nMAssay Description:Inverse agonist activity of LXRalpha (unknown origin)More data for this Ligand-Target Pair