Compile Data Set for Download or QSAR
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Found 3 of ic50 for monomerid = 17946
TargetRenin(Homo sapiens (Human))
Novartis Pharmaceuticals

LigandPNGBDBM17946((2S,4S,7R)-4-amino-7-(butylcarbamoyl)-5-hydroxy-2,...)
Affinity DataIC50:  3nMpH: 7.2 T: 2°CAssay Description:In vitro potencies of compounds against purified human recombinant renin were determined by its cleavage of substrate angiotensinogen. The angiotensi...More data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Novartis Pharmaceuticals

LigandPNGBDBM17946((2S,4S,7R)-4-amino-7-(butylcarbamoyl)-5-hydroxy-2,...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human reninMore data for this Ligand-Target Pair
TargetPepsin A(Porcine)
Novartis Pharmaceuticals

LigandPNGBDBM17946((2S,4S,7R)-4-amino-7-(butylcarbamoyl)-5-hydroxy-2,...)
Affinity DataIC50: >1.00E+5nMpH: 2.0 T: 2°CAssay Description:In vitro potencies of compounds against purified porcine pepsin were determined by its cleavage of substrate hemoglobin. After incubation, proteins w...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed