Affinity DataIC50: 0.330nMpH: 7.0Assay Description:In vitro inhibitory activity against porcine prolyl oligopeptidase by using 4 mM Suc-Gly-Pro-7-amido-4-methylcoumarin as substrate (pH 7.0) at 30 deg...More data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:In vitro inhibitory activity of the compound against prolyl oligopeptidase (POP) from pigbrain expressedMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:In vitro inhibitory activity against purified prolyl endopeptidase (PEP) from canine brain.More data for this Ligand-Target Pair
Affinity DataIC50: 1.27nMAssay Description:Inhibition of Flavobacterium meningosepticum propyl endopeptidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibition of POP (unknown origin) using (Z)-Gly-Pro-p-nitroanilide as substrate preincubated for 5 mins followed by substrate addition and measured ...More data for this Ligand-Target Pair
TargetChymotrypsin-like elastase family member 1(Homo sapiens (Human))
Kyungpook National University
Curated by ChEMBL
Kyungpook National University
Curated by ChEMBL
Affinity DataIC50: 51.6nMAssay Description:Inhibition of Flavobacterium meningosepticum PEPMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Inhibitory activity of the compound was evaluated against Post-proline cleaving enzyme from rat cortexMore data for this Ligand-Target Pair