Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ic50 for monomerid = 50226664
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Beijing University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50226664(2-hydroxy-3,9,10-trimethoxy-5,6-dihydroisoquino[3,...)
Affinity DataIC50:  470nMAssay Description:Inhibition of recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21 using H3K4me2 as substrate preincubated for 10 mins followed by su...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Beijing University Of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50226664(2-hydroxy-3,9,10-trimethoxy-5,6-dihydroisoquino[3,...)
Affinity DataIC50:  470nMAssay Description:Inhibition of recombinant KDM1A (unknown origin) expressed in Escherichia coli BL21 using H3K4Me2 peptide as substrate preincubated for 10 mins follo...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
National Cheng Kung University

Curated by ChEMBL
LigandPNGBDBM50226664(2-hydroxy-3,9,10-trimethoxy-5,6-dihydroisoquino[3,...)
Affinity DataIC50:  3.06E+4nMAssay Description:Inhibition of human CYP3A4 expressed in Escherichia coli assessed as inhibition of nifedipine oxidationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50226664(2-hydroxy-3,9,10-trimethoxy-5,6-dihydroisoquino[3,...)
Affinity DataIC50:  1.71E+5nMAssay Description:Inhibition of HIV1 RTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
University Of Illinois

Curated by ChEMBL
LigandPNGBDBM50226664(2-hydroxy-3,9,10-trimethoxy-5,6-dihydroisoquino[3,...)
Affinity DataIC50:  1.71E+5nMAssay Description:Inhibition of Human immunodeficiency virus 1 NL4.3 reverse transcriptase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed