Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ic50 for monomerid = 50241779
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50241779(CHEMBL4082159)
Affinity DataIC50:  200nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv N-terminal 6His-tagged LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50241779(CHEMBL4082159)
Affinity DataIC50:  216nMAssay Description:Inhibition of Mycobacterium tuberculosis LeuRS expressed in Escherichia coli Rosetta (DE3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50241779(CHEMBL4082159)
Affinity DataIC50:  1.32E+5nMAssay Description:Inhibition of human N-terminal 6His-tagged cytoplasmic LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorporation in to E...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine--tRNA ligase, mitochondrial(Homo sapiens)
Anacor Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50241779(CHEMBL4082159)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human N-terminal 6His-tagged mitochondrial LeuRS expressed in Escherichia coli BL21(DE3) assessed as L-[14C]leucine incorporation in to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed