TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Antagonist activity at LPA1 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 5(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 463nMAssay Description:Antagonist activity at LPA5 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 3(Homo sapiens (Human))
The University Of Memphis
Curated by ChEMBL
The University Of Memphis
Curated by ChEMBL
Affinity DataIC50: 752nMAssay Description:Antagonist activity at LPA3 receptor expressed in rat RH7777 cells assessed as inhibition of LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair