TargetYersiniabactin siderophore biosynthetic protein(Yersinia pestis CA88-4125)
Weill Medical College Of Cornell University
Curated by ChEMBL
Weill Medical College Of Cornell University
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of Yersinia pestis YbtE assessed as incorporation of [3H]salicyl group to HMWP2 proteinMore data for this Ligand-Target Pair
TargetSalicyl-AMP ligase / salicyl-S-ArCP synthetase(Mycobacterium tuberculosis)
Weill Medical College Of Cornell University
Curated by ChEMBL
Weill Medical College Of Cornell University
Curated by ChEMBL
Affinity DataIC50: 10.7nMAssay Description:Inhibition of adenylation activity of Mycobacterium tuberculosis MbtA after 30 mins by ATP-[32P]pyrophosphate exchange assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 2(Homo sapiens (Human))
University Of Bath
Curated by ChEMBL
University Of Bath
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human TRPM2 expressed in HEK293 cells assessed as inhibition of ADPR-induced maximum outward potassium current at +15 mV by wh...More data for this Ligand-Target Pair