Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ic50 for monomerid = 50430961
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430961(CHEMBL2337844)
Affinity DataIC50:  12nMAssay Description:Inhibition of trypsin-like activity of human constitutive 20s proteasome beta-2 subunit using Boc-LRR-AMC as substrate assessed as remaining activity...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430961(CHEMBL2337844)
Affinity DataIC50:  26nMAssay Description:Inhibition of chymotrypsin-like activity of human constitutive 20s proteasome beta-5 subunit using Suc-LLVY-AMC as substrate assessed as remaining ac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430961(CHEMBL2337844)
Affinity DataIC50:  370nMAssay Description:Inhibition of postacid activity of human constitutive 20s proteasome beta-1 subunit using Z-LLE-betaNA as substrate assessed as remaining activity in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Paris 6

Curated by ChEMBL
LigandPNGBDBM50430961(CHEMBL2337844)
Affinity DataIC50:  756nMAssay Description:Inhibition of chymotrypsin-like activity of proteasome beta-5 subunit in HEK293 cells using Suc-LLVY-Glo as substrate incubated for 2 hrs prior to su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed