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Found 17 of ic50 for monomerid = 50466843

Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))TBA

IC50: 17nMAssay Description:Inhibition of recombinant human DYRK1A expressed in Escherichia coli using DYRKtide peptide as substrate incubated for 110 mins in presence of ATP by...More data for this Ligand-Target Pair

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Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))TBA

BDBM50466843(CHEMBL4283240)

IC50: 24nMAssay Description:Inhibition of recombinant human DYRK1A expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scin...More data for this Ligand-Target Pair

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Dual specificity protein kinase CLK4(Homo sapiens (Human))TBA

BDBM50466843(CHEMBL4283240)

IC50: 24nMAssay Description:Inhibition of recombinant human CLK4 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scinti...More data for this Ligand-Target Pair

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Dual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))TBA

BDBM50466843(CHEMBL4283240)

IC50: 38nMAssay Description:Inhibition of recombinant human DYRK1B expressed in Sf9 insect cells using DYRKtide peptide as substrate incubated for 110 mins in presence of ATP by...More data for this Ligand-Target Pair

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Dual specificity protein kinase CLK1(Homo sapiens (Human))TBA

BDBM50466843(CHEMBL4283240)

IC50: 88nMAssay Description:Inhibition of recombinant human CLK1 expressed in Sf9 insect cells using myelin basic protein as substrate incubated for 110 mins in presence of ATP ...More data for this Ligand-Target Pair

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Dual specificity protein kinase CLK1(Homo sapiens (Human))TBA

BDBM50466843(CHEMBL4283240)

IC50: 158nMAssay Description:Inhibition of recombinant human CLK1 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scinti...More data for this Ligand-Target Pair

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Dual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))TBA

BDBM50466843(CHEMBL4283240)

IC50: 181nMAssay Description:Inhibition of GST-tagged DYRK1A (unknown origin) expressed in Escherichia coli DH5alpha using RRRFRPASPLRGPPK as substrate after 30 mins by kinase-gl...More data for this Ligand-Target Pair

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Dual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))TBA

BDBM50466843(CHEMBL4283240)

IC50: 185nMAssay Description:Inhibition of recombinant human DYRK1B expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scin...More data for this Ligand-Target Pair

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Dual specificity protein kinase CLK2(Homo sapiens (Human))TBA

BDBM50466843(CHEMBL4283240)

IC50: 630nMAssay Description:Inhibition of recombinant human CLK2 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scinti...More data for this Ligand-Target Pair

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Dual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))TBA

BDBM50466843(CHEMBL4283240)

IC50: 814nMAssay Description:Inhibition of recombinant human DYRK2 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scint...More data for this Ligand-Target Pair

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Dual specificity tyrosine-phosphorylation-regulated kinase 3(Homo sapiens (Human))TBA

BDBM50466843(CHEMBL4283240)

IC50: 1.22E+3nMAssay Description:Inhibition of recombinant human DYRK3 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scint...More data for this Ligand-Target Pair

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Dual specificity protein kinase CLK3(Homo sapiens (Human))TBA

BDBM50466843(CHEMBL4283240)

IC50: 4.92E+3nMAssay Description:Inhibition of recombinant human CLK3 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scinti...More data for this Ligand-Target Pair

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Dual specificity tyrosine-phosphorylation-regulated kinase 4(Homo sapiens (Human))TBA

BDBM50466843(CHEMBL4283240)

IC50: 8.37E+3nMAssay Description:Inhibition of recombinant human DYRK4 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric scint...More data for this Ligand-Target Pair

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Glycogen synthase kinase-3 beta(Homo sapiens (Human))TBA

BDBM50466843(CHEMBL4283240)

IC50: >1.00E+4nMAssay Description:Inhibition of recombinant human GSK-3beta expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric s...More data for this Ligand-Target Pair

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Casein kinase I isoform epsilon(Homo sapiens (Human))TBA

BDBM50466843(CHEMBL4283240)

IC50: >1.00E+4nMAssay Description:Inhibition of recombinant human CK1epsilon expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric ...More data for this Ligand-Target Pair

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Platelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))TBA

BDBM50466843(CHEMBL4283240)

IC50: >1.00E+4nMAssay Description:Inhibition of recombinant human CDK5/p25 expressed in Sf9 insect cells incubated for 60 mins in presence of ATP and [gamma33-P] ATP by radiometric sc...More data for this Ligand-Target Pair

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Amine oxidase [flavin-containing] A(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL

BDBM50466843(CHEMBL4283240)

IC50: >1.00E+4nMAssay Description:Inhibition of human recombinant MAO-A after 1 hr by by MAO-Glo assayMore data for this Ligand-Target Pair

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Filter my 17 hits

Targets 13▿
- Dual specificity tyrosine-phosphorylation-regulated kinase 1A 3
- Dual specificity protein kinase CLK1 2
- Dual specificity tyrosine-phosphorylation-regulated kinase 1B 2
- Platelet-derived growth factor receptor alpha/beta 1
- Amine oxidase [flavin-containing] A 1
- Dual specificity protein kinase CLK4 1
- Dual specificity protein kinase CLK3 1
- Dual specificity protein kinase CLK2 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 4 1
- Casein kinase I isoform epsilon 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 2 1
- Dual specificity tyrosine-phosphorylation-regulated kinase 3 1
- Glycogen synthase kinase-3 beta 1
Publications 1▿
- J Med Chem 61: 9791-9810 (2018) 2
Institutions 1▿
- Seoul National University 2
Affinity: 17 to 1.0E+4 nM▿
- IC50 17
- Affinity ≤ nM
Xtal structures: 1
Docked structures: 0
Catalog Cmpds: 0