Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ki for monomerid = 14746
LigandPNGBDBM14746((R)-6,7-Dimethoxy-4-[3-(4-trifluoromethoxy-phenoxy...)
Affinity DataKi:  185nM ΔG°:  -38.0kJ/molepH: 7.5 T: 2°CAssay Description:PDE activity was monitored by measuring the hydrolysis of [3H]-cAMP to [3H]-AMP using a scintillation proximity assay (SPA). [3H]-AMP was captured by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Homo sapiens (Human))
Pfizer

LigandPNGBDBM14746((R)-6,7-Dimethoxy-4-[3-(4-trifluoromethoxy-phenoxy...)
Affinity DataKi:  739nMAssay Description:PDE activity was monitored by measuring the hydrolysis of [3H]-cAMP to [3H]-AMP using a scintillation proximity assay (SPA). [3H]-AMP was captured by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3B(Homo sapiens (Human))
Pfizer

LigandPNGBDBM14746((R)-6,7-Dimethoxy-4-[3-(4-trifluoromethoxy-phenoxy...)
Affinity DataKi:  1.82E+3nMAssay Description:PDE activity was monitored by measuring the hydrolysis of [3H]-cAMP to [3H]-AMP using a scintillation proximity assay (SPA). [3H]-AMP was captured by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed