TargetcAMP-dependent protein kinase(Oryctolagus cuniculus (Rabbit))
University of California San Diego
University of California San Diego
Affinity DataKi: 11nM ΔG°: -46.2kJ/mole IC50: 18nMpH: 7.5 T: 2°CAssay Description:Cyclic AMP-dependent protein kinase (PKA) enzyme inhibition assay using purified recombinant C subunit of PKA (catalytic (C) subunit (cPKA)) with hol...More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nM ΔG°: -30.8kJ/mole IC50: 6.90E+3nMT: 2°CAssay Description:Protein kinase C (PKC) enzyme inhibition assay using purified rat brain protein kinase C from Calbiochem #539494.More data for this Ligand-Target Pair