Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ki for monomerid = 50013721
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50013721(8-Br-adenine | 8-Bromo-9H-purin-6-ylamine0.9M HCl ...)
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50013721(8-Br-adenine | 8-Bromo-9H-purin-6-ylamine0.9M HCl ...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50013721(8-Br-adenine | 8-Bromo-9H-purin-6-ylamine0.9M HCl ...)
Affinity DataKi: >3.00E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50013721(8-Br-adenine | 8-Bromo-9H-purin-6-ylamine0.9M HCl ...)
Affinity DataKi:  3.30E+4nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4-kinase type 2-alpha(Homo sapiens (Human))
Smith Kline & French Research

Curated by ChEMBL
LigandPNGBDBM50013721(8-Br-adenine | 8-Bromo-9H-purin-6-ylamine0.9M HCl ...)
Affinity DataKi:  1.48E+5nMAssay Description:Binding affinity (Ki) against human phosphatidylinositol 4-kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed