TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: >0.5nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]U-69593 as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 2.89nMAssay Description:Inhibition against Opioid receptor mu 1 using [3H]- DAMGO radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Research Triangle Institute
Curated by ChEMBL
Research Triangle Institute
Curated by ChEMBL
Affinity DataKi: >3nMAssay Description:Binding affinity towards Opioid receptor delta 1 using [3H]DADLE as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]DAMGO as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition against delta-opioid receptor using [3H]-DPDPE radioligand.More data for this Ligand-Target Pair