Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ki for monomerid = 50072441
TargetCoagulation factor X(Oryctolagus cuniculus)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  94nMAssay Description:Inhibition of serine protease factor Xa enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  94nMAssay Description:Inhibition of Factor XaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  94nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  94nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  480nMAssay Description:The binding affinity was measured towards human purified trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  480nMAssay Description:The compound was evaluated for inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  1.60E+4nMAssay Description:The binding affinity towards thrombin obtained from human purified enzymes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072441(CHEMBL323060 | CHEMBL92988 | [3-(3-Carbamimidoyl-p...)
Affinity DataKi:  1.60E+4nMAssay Description:The compound was evaluated for inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails Article