Affinity DataIC50: 0.240nMAssay Description:Compound was evaluated for the antagonistic activity against NK1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:Binding affinity against Neurokinin 1(NK1) receptor from human IM-9 cells using [I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 0.440nMAssay Description:Binding affinity against human NK2 receptors from HSKR-1 cells using [125I]-Iodohistidyl NKAMore data for this Ligand-Target Pair
Affinity DataIC50: 0.540nMAssay Description:Inverse agonist at human CB1 receptor expressed in SF9 cells assessed as decrease in GTPgammaS levelMore data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:Antagonism of the guinea pig tachykinin NK1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.35nMAssay Description:Inverse agonist at human CB1 receptor expressed in SF9 cells assessed as decrease in GTPgammaS levelMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Binding affinity for NK2 receptor in HSKR-1 cells was determined by using [125 I ]-Iodohistidyl NKA.More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Binding affinity for NK2 receptor in HSKR-1 cells was determined by using [125 I ]-Iodohistidyl NKA.More data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 2.5nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Compound was evaluated for the antagonistic activity against NK1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.07nMAssay Description:Inverse agonist at human CB1 receptor expressed in SF9 cells assessed as decrease in GTPgammaS levelMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Binding affinity for NK2 receptor in HSKR-1 cells was determined by using [125 I ]-Iodohistidyl NKA.More data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Binding affinity against Neurokinin 1(NK1) receptor from human IM-9 cells using [I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Binding affinity for NK2 receptor in HSKR-1 cells was determined by using [125 I ]-Iodohistidyl NKA.More data for this Ligand-Target Pair
Affinity DataIC50: 3.90nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity against human NK2 receptors from HSKR-1 cells using [125I]-Iodohistidyl NKAMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Displacement of [125I]-sauvagine from rat CRF-1 receptor expressed in human IMR-32 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 4.20nMAssay Description:Inverse agonist at human CB1 receptor expressed in SF9 cells assessed as decrease in GTPgammaS levelMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 4.5nMAssay Description:Binding affinity for NK2 receptor in HSKR-1 cells was determined by using [125 I ]-Iodohistidyl NKA.More data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Antagonistic activity against Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 5.30nMAssay Description:Antagonistic activity against Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 5.70nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Binding affinity for NK1 receptor in guinea pig lung was determined by using [125 I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Antagonistic activity against Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 5.90nMAssay Description:Antagonistic activity against Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMAssay Description:Displacement of [125I]-sauvagine from rat CRF-1 receptor expressed in human IMR-32 cells after 2 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20nMAssay Description:Antagonistic activity against Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataIC50: 6.20nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.20nMAssay Description:Binding affinity against Neurokinin 1(NK1) receptor from human IM-9 cells using [I]-Bolton Hunter labeled SPMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.30nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:Antagonistic activity against histamine H1 receptorMore data for this Ligand-Target Pair