Affinity DataKi: 150nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor of rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor of rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Displacement of [3H]R-PIA from adenosine A1 receptor of rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 680nMAssay Description:Displacement of [3H]PSB-11 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Affinity DataKi: 1.13E+3nMAssay Description:Displacement of [3H]-MSX-2 from Adenosine A2A receptor of rat striatal membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Warner-Lambert/Parke-Davis Pharmaceutical Research
Curated by PDSP Ki Database
Affinity DataKi: 1.18E+3nMAssay Description:Displacement of [3H]NECA from Adenosine A2A receptor of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8.20E+3nMAssay Description:Binding affinity towards human adenosine A2B receptor in VA13 fibroblasts as inhibition of adenylate cyclase at 10 uM; Less than 10% inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 1.39E+4nMAssay Description:Displacement of [3H]PSB-298 from human adenosine A2B receptor expressed in HEK293 cells at 10 uM; Less than 10% inhibitionMore data for this Ligand-Target Pair
Affinity DataKi: 7.00E+5nMAssay Description:Inhibitory constant towards indole N-methyl-transferaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+6nMAssay Description:Inhibition constant against Escherichia coli cyclopropane fatty acid synthaseMore data for this Ligand-Target Pair
Affinity DataKi: >5.40E+6nMAssay Description:Compound was tested for inhibition of Catechol O-methyltransferase using radiochemical assayMore data for this Ligand-Target Pair