Affinity DataEC50: 316nMAssay Description:Agonist activity at human FFA4 receptor expressed in U2OS cells assessed as calcium mobilization after 24 hrs by FLIPRMore data for this Ligand-Target Pair
Affinity DataEC50: 540nMAssay Description:Agonist activity at human GPR40 expressed in CHOK1 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataEC50: 540nMAssay Description:Agonist activity at GPR40 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+5nMAssay Description:Inhibition of human recombinant FAAHMore data for this Ligand-Target Pair
Affinity DataEC50: 4.80E+3nMAssay Description:Agonist activity at human GPR40 expressed in human HEK293 cells assessed as increase in intracellular calcium flux after 10 mins by fluorescence assa...More data for this Ligand-Target Pair
Affinity DataEC50: 4.80E+3nMAssay Description:Agonist activity at human FFA1 receptor expressed in HEK293 cells assessed as increase in intracellular Ca2+ flux by Fluo-4 dye based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+5nMAssay Description:Antagonist activity at histamine H3 receptor in electrically-stimulated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as calcium flux by FLIPR assayMore data for this Ligand-Target Pair