TargetDisintegrin and metalloproteinase domain-containing protein 17 [215-477,S266A,N452Q](Homo sapiens (Human))
Schering-Plough Research Institute
Schering-Plough Research Institute
Affinity DataKi: 0.0600nM ΔG°: -13.8kcal/molepH: 7.3 T: 2°CAssay Description:Enzyme activity was determined by a kinetic assay measuring the rate of increase in fluorescent intensity generated by the cleavage of an internally ...More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens
Curated by ChEMBL
University Of Athens
Curated by ChEMBL
Affinity DataKi: 0.560nMAssay Description:Inhibition of pig TACEMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens
Curated by ChEMBL
University Of Athens
Curated by ChEMBL
Affinity DataKi: 0.560nMAssay Description:Inhibition of porcine TACEMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Sus scrofa (pig))
University Of Athens
Curated by ChEMBL
University Of Athens
Curated by ChEMBL
Affinity DataKi: 0.560nMAssay Description:Affinity for Tumor necrosis factor alpha converting enzyme (TACE)More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 33(Homo sapiens (Human))
University Of Athens
Curated by ChEMBL
University Of Athens
Curated by ChEMBL
Affinity DataKi: 141nMAssay Description:Affinity for Matrix metalloprotease-3 (MMP-3)More data for this Ligand-Target Pair
Affinity DataKi: 141nMAssay Description:Binding affinity to MMP3More data for this Ligand-Target Pair
Affinity DataKi: 257nMAssay Description:Affinity for Matrix metalloprotease-8 (MMP-8)More data for this Ligand-Target Pair
TargetMatrilysin(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 259nMAssay Description:Binding affinity to MMP7More data for this Ligand-Target Pair
TargetMatrilysin(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 259nMAssay Description:Affinity for Matrix metalloprotease-7 (MMP-7)More data for this Ligand-Target Pair
TargetMatrilysin(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 1.42E+3nMAssay Description:Affinity for Matrix metalloprotease-13 (MMP-13)More data for this Ligand-Target Pair
Affinity DataKi: 1.42E+3nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
Affinity DataKi: 1.42E+3nMAssay Description:Binding affinity to MMP13More data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Inhibition of MMP16More data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Affinity for Matrix metalloprotease-16 (MMP-16)More data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 2.05E+3nMAssay Description:Binding affinity to MMP2More data for this Ligand-Target Pair
Target72 kDa type IV collagenase(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Target72 kDa type IV collagenase(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 2.05E+3nMAssay Description:Affinity for Matrix metalloprotease-2 (MMP-2)More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Affinity for Matrix metalloprotease-15 (MMP-15)More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Inhibition of MMP15More data for this Ligand-Target Pair
Affinity DataKi: 1.03E+4nMAssay Description:Affinity towards Matrix metalloprotease-9 (MMP-9)More data for this Ligand-Target Pair
Affinity DataKi: 1.59E+4nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
Affinity DataKi: 1.59E+4nMAssay Description:Affinity for Matrix metalloprotease-14 (MMP-14)More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+4nMAssay Description:Affinity towards Matrix metalloprotease-1 (MMP-1)More data for this Ligand-Target Pair