Affinity DataKi: 7.49E+3nM ΔG°: -7.27kcal/mole IC50: 3.48E+4nMpH: 7.4 T: 2°CAssay Description:Various concentrations of test compound (5, 10, 25, 50 and 100 mM) were dissolved in DMSO (final culture concentration 0.1%) and 4-MU oleate and lipa...More data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of Louisiana At Monroe
Curated by ChEMBL
University Of Louisiana At Monroe
Curated by ChEMBL
Affinity DataIC50: 2.02E+4nMAssay Description:Inhibition of recombinant human N-terminal His-tagged cytoplasmic c-MET kinase domain (956 to 1390 residues) phosphorylation expressed in baculovirus...More data for this Ligand-Target Pair