Affinity DataKi: 0.300nMAssay Description:In vitro inhibitory constant against [125I]DOI binding to 5-hydroxytryptamine 2A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibitory constant against cloned human 5-hydroxytryptamine 2A receptor using with [125I]- DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Inhibitory constant against cloned human 5-hydroxytryptamine 2C receptor using with [125I]- DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibitory constant against cloned human 5-hydroxytryptamine 2B receptor using with [125I]- DOI radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Inhibitory constant against human 5-hydroxytryptamine 6 receptor using [3H]LSD radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Inhibitory constant against 5-hydroxytryptamine 4 receptor using [3H]GR-113808 radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Inhibitory constant against human 5-hydroxytryptamine 5A receptor using [3H]LSD radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory constant against 5-hydroxytryptamine 3 receptor using [3H]GR-65630 radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory constant against human serotonin transporter using [3H]N-Me-citalopram radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory constant against 5-hydroxytryptamine 1B receptor using with [125I]- cyanopindolol radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory constant against human 5-hydroxytryptamine 1B receptor using [3H]5-CT radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Inhibitory constant against Alpha-2B adrenergic receptor using [3H]MK-912 radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+4nMAssay Description:Inhibitory constant against human 5-hydroxytryptamine 7 receptor using [3H]LSD radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+4nMAssay Description:Inhibitory constant against Alpha-1B adrenergic receptor using [3H]-7-MeO prazosin radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Alcon Research
Curated by ChEMBL
Alcon Research
Curated by ChEMBL
Affinity DataKi: >3.00E+4nMAssay Description:Inhibitory constant against norepinephrine transporter receptor using [3H]radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >3.00E+4nMAssay Description:Inhibitory constant against Alpha-1A adrenergic receptor using [3H]-7-MeO prazosin radioligandMore data for this Ligand-Target Pair