Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ic50 for monomerid = 50154842
TargetCytochrome P450 3A4(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50154842(CHEMBL3775589 | US10273244, Example 12 | US1058413...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human CYP3A4 expressed in baculosomes preincubated for 10 mins followed by cofactor addition measured every minute for 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50154842(CHEMBL3775589 | US10273244, Example 12 | US1058413...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human CYP2D6 expressed in baculosomes preincubated for 10 mins followed by cofactor addition measured every minute for 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50154842(CHEMBL3775589 | US10273244, Example 12 | US1058413...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human CYP3A4 expressed in baculosomes preincubated for 10 mins followed by cofactor addition measured every minute for 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50154842(CHEMBL3775589 | US10273244, Example 12 | US1058413...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human CYP2C9 expressed in baculosomes preincubated for 10 mins followed by cofactor addition measured every minute for 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50154842(CHEMBL3775589 | US10273244, Example 12 | US1058413...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human CYP2C19 expressed in baculosomes preincubated for 10 mins followed by cofactor addition measured every minute for 10 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50154842(CHEMBL3775589 | US10273244, Example 12 | US1058413...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant human CYP1A2 expressed in baculosomes preincubated for 10 mins followed by cofactor addition measured every minute for 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50154842(CHEMBL3775589 | US10273244, Example 12 | US1058413...)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of human ERG tail current expressed in HEK293 cells after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50154842(CHEMBL3775589 | US10273244, Example 12 | US1058413...)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of human ERG tail current expressed in HEK293 cells after 5 mins by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed