Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ec50 for monomerid = 50245587
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50245587(CHEMBL4077064 | US10000483, Compound II-4)
Affinity DataEC50:  475nMAssay Description:Inhibition of 3x-FLAG-tagged BTK (unknown origin) expressed in HEK293T cells assessed as reduction in enzyme autophosphorylation at Y551 residue incu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50245587(CHEMBL4077064 | US10000483, Compound II-4)
Affinity DataEC50:  318nMAssay Description:Inhibition of BTK in human Ramos cells assessed as reduction in PLCgamma2 phosphorylation at Tyr759 residue by chemiluminescence based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed