Compile Data Set for Download or QSAR
maximum 50k data
Found 18 of ic50 for monomerid = 50269556
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of recombinant full-length His6-tagged BTK (unknown origin) expressed in baculovirus infected Sf9 cells using biotinylated A5 peptide as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  26nMAssay Description:Inhibition of BTK in human PBMC assessed as reduction in anti-IgM-induced MIP1betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  100nMAssay Description:Inhibition of LCK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Srms(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  103nMAssay Description:Inhibition of SRMS (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine kinase 6(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  173nMAssay Description:Inhibition of PTK6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Yes(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  266nMAssay Description:Inhibition of YES1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fgr(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  268nMAssay Description:Inhibition of FGR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Blk(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  280nMAssay Description:Inhibition of BLK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  428nMAssay Description:Inhibition of TEC (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase TXK(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  464nMAssay Description:Inhibition of TXK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  512nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  514nMAssay Description:Inhibition of ERBB4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  703nMAssay Description:Inhibition of BMX (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase FRK(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  706nMAssay Description:Inhibition of FRK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of LYNB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of FYN (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase CSK(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  2.15E+3nMAssay Description:Inhibition of CSK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50269556(CHEMBL4075954)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human ERG by [35S]-MK499 displacement or iKr channel assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed