Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of ki for monomerid = 50359391
TargetVesicular acetylcholine transporter(Rattus norvegicus)
Iqog, Csic

Curated by ChEMBL
LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataKi:  2.60nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in rat PC12 cell membranes after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Iqog, Csic

Curated by ChEMBL
LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataKi:  2.80nMAssay Description:Displacement of (+)-[3H]pentazocine from human sigma1 receptor expressed in HEK293 cell membranes after 60 mins by liquid scintillation counting meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataKi:  11nMAssay Description:Non-competitive inhibition of rat liver mitochondrial MAO-B using phenylethylamine as substrate by Line-Weaver Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
Iqog, Csic

Curated by ChEMBL
LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]DTG from sigma2 receptor in rat liver membranes after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataKi:  84nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Julius Maximilian University Of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human H3R expressed in HEK293 cell membranes incubated for 90 mins by liquid scintillation counting...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Universitat Aut£Noma De Barcelona

Curated by ChEMBL
LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataKi:  149nMAssay Description:Mixed type inhibition of Electrophorus electricus AchE using acetylthiocholine as substrate by Line-Weaver Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed