Compile Data Set for Download or QSAR
Report error Found 7 of ec50 for monomerid = 50378072
TargetBeta-3 adrenergic receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378072BDBM50378072(CHEMBL1204383)
Affinity DataEC50:  1.60nMAssay Description:Agonistic activity was assessed by measuring cAMP accumulation in CHO cell lines expressing cloned human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378072BDBM50378072(CHEMBL1204383)
Affinity DataEC50:  3.60nMAssay Description:Agonistic activity was assessed by measuring cAMP accumulation in CHO cell lines expressing cloned human Beta-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378072BDBM50378072(CHEMBL1204383)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human cloned adrenergic beta-1 receptor expressed in CHO cells assessed as [125I]cAMP accumulation after 2 days by radioimmunoass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378072BDBM50378072(CHEMBL1204383)
Affinity DataEC50:  380nMAssay Description:Agonist activity at human cloned adrenergic beta3 receptor expressed in CHO cells assessed as [125I]cAMP accumulation after 2 days by radioimmunoassa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378072BDBM50378072(CHEMBL1204383)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human cloned adrenergic beta3 receptor expressed in CHO cells assessed as [125I]cAMP accumulation after 2 days by radioimmunoassa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378072BDBM50378072(CHEMBL1204383)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human cloned adrenergic beta-1 receptor expressed in CHO cells assessed as [125I]cAMP accumulation after 2 days by radioimmunoass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Astellas Pharma

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50378072BDBM50378072(CHEMBL1204383)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human cloned adrenergic beta2 receptor expressed in CHO cells assessed as [125I]cAMP accumulation after 2 days by radioimmunoassa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed