Affinity DataIC50: 0.0270nMAssay Description:Binding affinity against human Melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0300nMAssay Description:Binding affinity against human Melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0600nMAssay Description:Binding affinity against human Melanocortin-4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Binding affinity against human Melanocortin-4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Binding affinity against human Melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Binding affinity against human Melanocortin 5 receptorMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Displacement of [125I]NDPalphaMSH from human cloned melanocortin receptor 1b expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Displacement of [125I]NDPalphaMSH from human cloned MC4R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Displacement of [125I]NDPalphaMSH from human cloned MC5R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Binding affinity against human Melanocortin-4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.190nMAssay Description:Binding affinity for human Melanocortin-3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.210nMAssay Description:Binding affinity for human Melanocortin-3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.230nMAssay Description:Binding affinity for human Melanocortin-3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.230nMAssay Description:Binding affinity against human Melanocortin-4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Evaluated for binding affinity against Melanocortin-4 receptor by displacing [125I]-NDP-alpha-MSH radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMAssay Description:Concentration required for 50% inhibition by displacement of of [125I]NDP-alpha-MSH of human MC4R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.410nMAssay Description:Inhibition of human MC4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Inhibition of human MC4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.480nMAssay Description:Binding affinity against human Melanocortin-4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against human Melanocortin-4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Binding affinity to rat MC4RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Evaluated for binding affinity against Melanocortin-4 receptor by displacing [125I]-NDP-alpha-MSH radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.510nMAssay Description:Binding affinity against human Melanocortin-4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.530nMAssay Description:Displacement of [125I]-NDP-R-MSH from human MC4R expressed in CHO cells after 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:Concentration required for 50% inhibition by displacement of of [125I]NDP-alpha-MSH of human MC4R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Evaluated for binding affinity against rat Melanocortin-4 receptor (rMC4R) by displacing [125I]NDP-alpha-MSH radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.620nMAssay Description:Activity against human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.710nMAssay Description:Displacement of [125I]-NDP-R-MSH from human MC4R expressed in CHO cells after 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.770nMAssay Description:Concentration required for 50% inhibition by displacement of of [125I]NDP-alpha-MSH of human MC4R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.780nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Activity against human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.840nMAssay Description:Inhibition of human MC4 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.850nMAssay Description:Displacement of [125I]-NDP-R-MSH from human MC4R expressed in CHO cells after 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.850nMAssay Description:Binding affinity to human MC4RMore data for this Ligand-Target Pair
Affinity DataIC50: 0.890nMAssay Description:Binding affinity for Human Melanocortin 5 receptor expressed in L-cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.890nMAssay Description:Displacement of [125I]-NDP-R-MSH from human MC4R expressed in CHO cells after 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human melanocortin 4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.910nMAssay Description:Activity against human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.950nMAssay Description:Displacement of [125I]NDPalphaMSH from human cloned MC5R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human melanocortin 4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity to rat MC4RMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]-NDP-R-MSH from human MC4R expressed in CHO cells after 1.5 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Concentration required for 50% inhibition by displacement of of [125I]NDP-alpha-MSH of human MC4R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Concentration required for 50% inhibition by displacement of of [125I]NDP-alpha-MSH of human MC4R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Binding affinity against human Melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Activity against human MC4R by cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Evaluated for binding affinity against Melanocortin-4 receptor by displacing [125I]-NDP-alpha-MSH radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Evaluated for binding affinity against human Melanocortin-4 receptor (hMC4R) by displacing [125I]-NDP-alpha-MSH radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Concentration required to inhibit binding of [125I]-NDP-alpha-MSH from membranes prepared from CHO cells expressing human melanocortin subtype-4-rece...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Evaluated for Functional Activity at Melanocortin-4 receptor as effective concentration at 50% maximum CMP accumulationMore data for this Ligand-Target Pair