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Found 8 of ic50 for UniProtKB: P34903
LigandPNGBDBM50608946(CHEMBL2008708)
Affinity DataIC50:  16nMAssay Description:Inhibition of GABAA alpha3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand Info
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LigandPNGBDBM50608947(CHEMBL5281056)
Affinity DataIC50:  31nMAssay Description:Inhibition of GABAA alpha3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand Info
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TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50588336(CHEMBL5186739)
Affinity DataIC50:  79nMAssay Description:Antagonist activity at human alpha3beta2gamma2 GABAA receptor expressed in HEKcells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50588337(CHEMBL5177970)
Affinity DataIC50:  288nMAssay Description:Antagonist activity at human alpha3beta2gamma2 GABAA receptor expressed in HEKcells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50588339(CHEMBL5187612)
Affinity DataIC50:  501nMAssay Description:Antagonist activity at human alpha3beta2gamma2 GABAA receptor expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50329649(1-phenylethyl 9H-pyrido[3,4-b]indole-3-carboxylate...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human recombinant GABAA alpha3 receptorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50588340(CHEMBL5204910)
Affinity DataIC50:  3.24E+3nMAssay Description:Antagonist activity at human alpha3beta2gamma2 GABAA receptor expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50580362(CHEMBL5086854)
Affinity DataIC50:  5.50E+3nMAssay Description:Negative allosteric modulation activity at human GABAA alpha3beta3gamma2 stably expressed in HEK cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed