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Found 25 of ic50 for UniProtKB: P47211
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50208989(CHEMBL506553)
Affinity DataIC50:  0.0790nMAssay Description:Displacement of [125I]galanin from human recombinant GAL1 receptor expressed in HEK293 cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataIC50:  0.160nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50378616(GALANIN)
Affinity DataIC50:  0.770nMAssay Description:Binding affinity to human GAL1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358662(CHEMBL1922003)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358673(CHEMBL1922025)
Affinity DataIC50:  2.82E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358659(CHEMBL1922000)
Affinity DataIC50:  3.35E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358669(CHEMBL1922021)
Affinity DataIC50:  3.84E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358670(CHEMBL1922022)
Affinity DataIC50:  3.84E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358660(CHEMBL1922001)
Affinity DataIC50:  3.90E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358653(CHEMBL1921993)
Affinity DataIC50:  4.60E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358655(CHEMBL1921996)
Affinity DataIC50:  5.03E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358667(CHEMBL1922016)
Affinity DataIC50:  5.48E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358657(CHEMBL1921998)
Affinity DataIC50:  5.62E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358656(CHEMBL1921997)
Affinity DataIC50:  5.93E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358661(CHEMBL1922002)
Affinity DataIC50:  6.32E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358651(CHEMBL1921991)
Affinity DataIC50:  6.77E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358668(CHEMBL1922019)
Affinity DataIC50:  6.78E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358658(CHEMBL1921999)
Affinity DataIC50:  6.82E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358671(CHEMBL1922023)
Affinity DataIC50:  6.82E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358650(CHEMBL1921989)
Affinity DataIC50:  6.90E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358648(CHEMBL1921902)
Affinity DataIC50:  8.59E+3nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358652(CHEMBL1921992)
Affinity DataIC50:  1.28E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358672(CHEMBL1922024)
Affinity DataIC50:  1.60E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358654(CHEMBL1921995)
Affinity DataIC50:  2.75E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 1(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50358649(CHEMBL1921903)
Affinity DataIC50:  3.49E+4nMAssay Description:Displacement of [125I]galanin from GalR1 by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed