Compile Data Set for Download or QSAR
maximum 50k data
Found 13 of ic50 for UniProtKB: Q8VH26
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595404(CHEMBL5184455)
Affinity DataIC50:  0.100nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595426(CHEMBL5193853)
Affinity DataIC50:  0.126nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595424(CHEMBL5172865)
Affinity DataIC50:  0.200nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595403(CHEMBL5208201)
Affinity DataIC50:  0.200nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595425(CHEMBL5208957)
Affinity DataIC50:  0.398nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50296345((1R,2R,4S,5R,7S)-7-(2-hydroxy-2,2-di-thiophen-2-yl...)
Affinity DataIC50:  0.410nMAssay Description:Antagonist activity at M3 receptor in Dunkin-Hartley guinea pig tracheal strips assessed as inhibition of electrically field-stimulated contractile r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595423(CHEMBL5190387)
Affinity DataIC50:  0.501nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50355622(CHEMBL1910856)
Affinity DataIC50:  1.53nMAssay Description:Antagonist activity at M3 receptor in Dunkin-Hartley guinea pig tracheal strips assessed as inhibition of electrically field-stimulated contractile r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595427(CHEMBL5200887)
Affinity DataIC50:  2nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50355631(CHEMBL1910865)
Affinity DataIC50:  3.48nMAssay Description:Antagonist activity at M3 receptor in Dunkin-Hartley guinea pig tracheal strips assessed as inhibition of electrically field-stimulated contractile r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50355616(CHEMBL1910850)
Affinity DataIC50:  3.87nMAssay Description:Antagonist activity at M3 receptor in Dunkin-Hartley guinea pig tracheal strips assessed as inhibition of electrically field-stimulated contractile r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50355617(CHEMBL1910851)
Affinity DataIC50:  4.30nMAssay Description:Antagonist activity at M3 receptor in Dunkin-Hartley guinea pig tracheal strips assessed as inhibition of electrically field-stimulated contractile r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor(Cavia porcellus)
Chiesi Farmaceutici

Curated by ChEMBL
LigandPNGBDBM50595405(CHEMBL5184598)
Affinity DataIC50:  7.90nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed