Affinity DataKi: 43nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of Dengue virus serotype 2 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of Dengue virus serotype 1 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of Dengue virus serotype 1 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Inhibition of Dengue virus serotype 2 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Inhibition of Dengue virus serotype 1 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Inhibition of Dengue virus serotype 1 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Inhibition of Dengue virus serotype 2 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:Inhibition of Dengue virus serotype 2 NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Nle-Lys-Arg-Arg-Ser-3-(NO2)Ty...More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of Dengue virus serotype 3 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Inhibition of Dengue virus serotype 3 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Inhibition of Dengue virus serotype 3 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 665nMAssay Description:Binding affinity to DENV NS2B-NS3 protease assessed as inhibition constant using benzoyl-Nle-Lys-Arg-Arg-AMC as substrate incubated for 60 min by mea...More data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Inhibition of Dengue virus serotype 3 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 750nMAssay Description:Non-competitive inhibition of Dengue virus 3 NS3 helicaseMore data for this Ligand-Target Pair
Affinity DataKi: 750nMAssay Description:Non-competitive inhibition of Dengue virus 4 NS3 helicaseMore data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of Dengue virus serotype 2 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Inhibition of Dengue virus serotype 4 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Inhibition of Dengue virus serotype 4 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Inhibition of Dengue virus serotype 4 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 2.70E+3nMAssay Description:Inhibition of Dengue virus serotype 4 NS2B-NS3 protease preincubated for 20 mins followed by Abz-RRRRSAG-nY-NH2 addition and measured for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+3nMAssay Description:Competitive inhibition of DENV2 NS2B-NS3 protease expressed in Escherichia coli BL21 lambda(DE3) using FRET substrate preincubated with enzyme for 15...More data for this Ligand-Target Pair
Affinity DataKi: 3.80E+3nMAssay Description:Inhibition of Dengue virus serotype 2 NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells using Abz-Nle-Lys-Arg-Arg-Ser-3-(NO2)Ty...More data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nMAssay Description:Competitive inhibition of DENV2 NS2B-NS3 protease expressed in Escherichia coli BL21 lambda(DE3) using FRET substrate preincubated with enzyme for 15...More data for this Ligand-Target Pair
Affinity DataKi: 4.20E+3nMAssay Description:Inhibition of Dengue virus 1 NS2B-NS3 protease expressed in Escherichia coli using Abz-RRRRSAG-nY-NH2 as substrate preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Affinity DataKi: 4.80E+3nMAssay Description:Inhibition of Dengue virus 2 NS2B-NS3 protease expressed in Escherichia coli using Abz-RRRRSAG-nY-NH2 as substrate preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Affinity DataKi: 4.90E+3nMAssay Description:Inhibition of Dengue virus serotype 2 NS2B-NS3 protease preincubated for 15 mins followed by Abz-Nle-Lys-Arg-Arg-Ser-3-(NO2)Tyr addition and measured...More data for this Ligand-Target Pair
Affinity DataKi: 4.90E+3nMAssay Description:Inhibition of Dengue virus 2 NS2B-NS3 protease using Abz-Nle-Lys-Arg-Arg-Ser-3-(NO2)Tyr as substrate preincubated for 15 mins followed by addition of...More data for this Ligand-Target Pair
Affinity DataKi: 5.20E+3nMAssay Description:Competitive inhibition of DENV2 NS2B-NS3 protease expressed in Escherichia coli BL21 lambda(DE3) using FRET substrate preincubated with enzyme for 15...More data for this Ligand-Target Pair
Affinity DataKi: 5.30E+3nMAssay Description:Binding affinity to DENV2 NS2B/NS3 protease assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 5.30E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 5.30E+3nMAssay Description:Inhibition of DENV2 NS2B-NS3 proteaseMore data for this Ligand-Target Pair
Affinity DataKi: 5.80E+3nMAssay Description:Inhibitory activity against CF40.NS3pro from Dengue virus type 2More data for this Ligand-Target Pair
Affinity DataKi: 5.80E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 6.10E+3nMAssay Description:Competitive inhibition of DENV2 NS2B-NS3 protease expressed in Escherichia coli BL21 lambda(DE3) using FRET substrate preincubated with enzyme for 15...More data for this Ligand-Target Pair
Affinity DataKi: 6.30E+3nMAssay Description:Competitive inhibition of DENV2 NS2B-NS3 protease expressed in Escherichia coli BL21 lambda(DE3) using FRET substrate preincubated with enzyme for 15...More data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 6.90E+3nMAssay Description:Competitive inhibition of DENV2 NS2B-NS3 protease expressed in Escherichia coli BL21 lambda(DE3) using FRET substrate preincubated with enzyme for 15...More data for this Ligand-Target Pair
Affinity DataKi: 7.00E+3nMAssay Description:Mixed noncompetitive inhibition of the Dengue virus 2 NS2B-NS3 protease expressed in Escherichia coli using Boc-GRR-AMC as substrate assessed as enzy...More data for this Ligand-Target Pair
Affinity DataKi: 7.25E+3nMAssay Description:Binding affinity to DENV NS2B-NS3 protease assessed as inhibition constant using benzoyl-Nle-Lys-Arg-Arg-AMC as substrate incubated for 60 min by mea...More data for this Ligand-Target Pair
Affinity DataKi: 7.50E+3nMAssay Description:Inhibitory activity against dengue 2 NS3 protease fused via a linker to region of NS2BMore data for this Ligand-Target Pair
Affinity DataKi: 7.67E+3nMAssay Description:Binding affinity to DENV2 NS2B-NS3 protease by Dixon plot analysisMore data for this Ligand-Target Pair