Compile Data Set for Download or QSAR
maximum 50k data
Found 52 of ec50 for UniProtKB: P32301
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50604669(CHEMBL5208485)
Affinity DataEC50:  0.00800nMAssay Description:Positive allosteric modulator activity at GLP-1R in rat INS1 beta-cells assessed potentiation of GLP-1(7-36)NH2 induced insulin secretion incubated f...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393580(CHEMBL2158410)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50557261(CHEMBL4749279)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at rat GLP-1R expressed in HEK293 cells assessed as stimulation of cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50604669(CHEMBL5208485)
Affinity DataEC50:  0.25nMAssay Description:Positive allosteric modulator activity at GLP-1R in rat INS1 beta-cells assessed potentiation of GLP-1(7-36)NH2 induced insulin secretion incubated f...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50231948(CHEMBL4066463)
Affinity DataEC50:  0.25nMAssay Description:Agonist activity at GLP1R in rat INS-1 cells assessed as increase in glucose-stimulated insulin secretion after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50557264(CHEMBL4751466)
Affinity DataEC50:  0.480nMAssay Description:Agonist activity at rat GLP-1R expressed in HEK293 cells assessed as stimulation of cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50261506(CHEMBL499930 | HAEGTFTSDVSSYLEGQAAKEFIAWLVKGRG-NH2)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at GLP1R in rat INS-1 cells assessed as increase in glucose-stimulated insulin secretion after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50231943(CHEMBL4093072)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at GLP1R in rat INS-1 cells assessed as increase in glucose-stimulated insulin secretion after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50231901(CHEMBL4088708)
Affinity DataEC50:  16nMAssay Description:Agonist activity at GLP1R in rat INS-1 cells assessed as increase in glucose-stimulated insulin secretion after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50231886(CHEMBL4070761)
Affinity DataEC50:  50nMAssay Description:Agonist activity at GLP1R in rat INS-1 cells assessed as increase in glucose-stimulated insulin secretion after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393574(CHEMBL2158422)
Affinity DataEC50:  118nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50231963(CHEMBL4104146)
Affinity DataEC50:  130nMAssay Description:Agonist activity at GLP1R in rat INS-1 cells assessed as increase in glucose-stimulated insulin secretion after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393576(CHEMBL2158419)
Affinity DataEC50:  148nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393572(CHEMBL2158488)
Affinity DataEC50:  203nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393590(CHEMBL2158404)
Affinity DataEC50:  326nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50260246(1,3-bis(4-(tert-butoxycarbonyl)benzamido)-2,4-bis(...)
Affinity DataEC50:  370nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50260246(1,3-bis(4-(tert-butoxycarbonyl)benzamido)-2,4-bis(...)
Affinity DataEC50:  371nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50260245(1,3-bis(4-(cyclopentanecarboxamido)benzamido)-2,4-...)
Affinity DataEC50:  657nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393573(CHEMBL2158423)
Affinity DataEC50:  696nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393575(CHEMBL2158420)
Affinity DataEC50:  749nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50260245(1,3-bis(4-(cyclopentanecarboxamido)benzamido)-2,4-...)
Affinity DataEC50:  1.08E+3nMAssay Description:Agonist activity at rat GLP1 receptor expressed in HEK293 cells assessed as cAMP releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393571(CHEMBL2158489)
Affinity DataEC50:  1.11E+3nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393586(CHEMBL2158409)
Affinity DataEC50:  1.38E+3nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393568(CHEMBL2158495)
Affinity DataEC50:  2.13E+3nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393585(CHEMBL2158311)
Affinity DataEC50:  2.15E+3nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393588(CHEMBL2158407)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393567(CHEMBL2158496)
Affinity DataEC50:  2.71E+3nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50260246(1,3-bis(4-(tert-butoxycarbonyl)benzamido)-2,4-bis(...)
Affinity DataEC50:  2.73E+3nMAssay Description:Agonist activity at rat GLP1 receptor expressed in HEK293 cells assessed as cAMP releaseMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393587(CHEMBL2158408)
Affinity DataEC50:  3.33E+3nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393570(CHEMBL2158492)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393566(CHEMBL2158497)
Affinity DataEC50:  4.50E+3nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393589(CHEMBL2158406)
Affinity DataEC50:  8.31E+3nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393569(CHEMBL2158494)
Affinity DataEC50:  9.12E+3nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393598(CHEMBL2158393)
Affinity DataEC50:  9.40E+3nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393581(CHEMBL2158316)
Affinity DataEC50:  1.58E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393583(CHEMBL2158313)
Affinity DataEC50:  1.91E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393577(CHEMBL2158417)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393565(CHEMBL2158391)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM349662(2-{[4-(6-{[(4-cyano-2-fluorophenyl)(methyl-d2)]oxy...)
Affinity DataEC50: >2.00E+4nMAssay Description:Activation of rat GLP-1R expressed in CHO cells assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393564(CHEMBL2158392)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393578(CHEMBL2158416)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393579(CHEMBL2158415)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50260246(1,3-bis(4-(tert-butoxycarbonyl)benzamido)-2,4-bis(...)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393597(CHEMBL2158394)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393596(CHEMBL2158395)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393595(CHEMBL2158397)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393594(CHEMBL2158399)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393593(CHEMBL2158400)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393592(CHEMBL2158401)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Rattus norvegicus)
Hospital Regional Universitario

Curated by ChEMBL
LigandPNGBDBM50393591(CHEMBL2158402)
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at rat GLP1R expressed in HEK293 cells assessed as stimulation of cAMP levels incubated for 6 hrs by multiple response element/cAMP ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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