Affinity DataKi: 0.380nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 0.630nMAssay Description:Inhibition of [3H]PDBu binding to PKC gamma C1A peptideMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Displacement of 3H-PDBu from recombinant human PKCgamma incubated for 25 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domain (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC gamma expressed in baculovirusMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibition of human Protein kinase C gamma with [Ca2+]More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C eta C1a domainMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C eta C1a domainMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C gammaMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
Affinity DataKi: 19.4nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC gamma expressed in baculovirusMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of 3H-PDBu from recombinant human PKCgamma incubated for 25 mins by scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Inhibition of [3H]PDBu binding to PKC gamma C1A peptideMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 40.7nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC gamma expressed in baculovirusMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C gammaMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Inhibition of [3H]PDBu binding to PKC gamma C1A peptideMore data for this Ligand-Target Pair
TargetO94806/P05129/P05771/P17252/P24723/P41743/Q02156/Q04759/Q05513/Q05655/Q15139(Homo sapiens (Human))
Ura Cnrs 1309
Curated by ChEMBL
Ura Cnrs 1309
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Displacement of ATP from protein kinase C (PKC)More data for this Ligand-Target Pair
Affinity DataKi: 138nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
Affinity DataKi: 138nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to Protein kinase C eta C1a domainMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC gamma expressed in baculovirusMore data for this Ligand-Target Pair
Affinity DataKi: 151nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/gamma/delta/epsilon/eta/theta type/Serine/threonine-protein kinase D1/D3(Homo sapiens (Human))
National Cancer Institute-Frederick
Curated by ChEMBL
National Cancer Institute-Frederick
Curated by ChEMBL
Affinity DataKi: 190nMAssay Description:Displacement of [3H]PDBu binding to Protein kinase C of CEM cells with 10% fetal calf serumMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/gamma/delta/epsilon/eta/theta type/Serine/threonine-protein kinase D1/D3(Homo sapiens (Human))
National Cancer Institute-Frederick
Curated by ChEMBL
National Cancer Institute-Frederick
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase CMore data for this Ligand-Target Pair
Affinity DataKi: 209nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C gammaMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Inhibition of PKCgamma (unknown origin)More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/gamma/delta/epsilon/eta/theta type/Serine/threonine-protein kinase D1/D3(Homo sapiens (Human))
National Cancer Institute-Frederick
Curated by ChEMBL
National Cancer Institute-Frederick
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Displacement of [3H]PDBu from Protein kinase C of CEM cellsMore data for this Ligand-Target Pair
Affinity DataKi: 213nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C gamma C1b domainMore data for this Ligand-Target Pair
Affinity DataKi: 213nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
Affinity DataKi: 225nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
Affinity DataKi: 234nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
Affinity DataKi: 279nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C gammaMore data for this Ligand-Target Pair