Affinity DataIC50: 5.10nMAssay Description:Inhibition of steroid sulfatase in human JEG3 cell using [3H] E1S as substrate after 1 hr by scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Inhibition of steroid sulfatase in human JEG3 cell using [3H] E1S as substrate after 1 hr by scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of steroid sulfatase in human JEG3 cell using [3H] E1S as substrate after 1 hr by scintillation spectrometry analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate preincubated for 10 mins at pH 8More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of steroid sulfatase in human JEG3 cell using [3H] E1S as substrate after 1 hr by scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of steroid sulfatase in human JEG3 cell using [3H] E1S as substrate after 1 hr by scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibition of steroid sulfatase in human JEG3 cell using [3H] E1S as substrate after 1 hr by scintillation spectrometry analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate preincubated for 10 mins at pH 6More data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Inhibition of steroid sulfatase in human JEG3 cell using [3H] E1S as substrate after 1 hr by scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Inhibition of steroid sulfatase in human JEG3 cell using [3H] E1S as substrate after 1 hr by scintillation spectrometry analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 135nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 139nMAssay Description:Inhibition of steroid sulfatase in human JEG3 cell using [3H] E1S as substrate after 1 hr by scintillation spectrometry analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 331nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 589nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Inhibition of FAAH (unknown origin) expressed in human HeLa cells transfected with empty vector using [3H]AEA as substrate after 2 hrs by liquid scin...More data for this Ligand-Target Pair
Affinity DataIC50: 700nMAssay Description:Inhibition of FAAH (unknown origin) expressed in human HeLa cells using [3H]AEA as substrate after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 740nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 741nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 990nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of steroid sulfatase in human JEG3 cell using [3H] E1S as substrate after 1 hr by scintillation spectrometry analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.69E+3nMAssay Description:Inhibition of steroid sulfatase in human JEG3 cell using [3H] E1S as substrate after 1 hr by scintillation spectrometry analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of FAAH T488A mutant (unknown origin) expressed in human HeLa cells using [3H]AEA as substrate after 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of FAAH T488A mutant (unknown origin) expressed in human HeLa cells using [3H]AEA as substrate after 2 hrs by liquid scintillation countin...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of FAAH (unknown origin) expressed in human HeLa cells using [3H]AEA as substrate after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of FAAH (unknown origin) expressed in human HeLa cells transfected with empty vector using [3H]AEA as substrate after 2 hrs by liquid scin...More data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 3.09E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 4.27E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
University Of Cagliari
Curated by ChEMBL
University Of Cagliari
Curated by ChEMBL
Affinity DataIC50: 6.46E+3nMAssay Description:Inhibition of rat brain FAAH using [3H]AEA as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of FAAH (unknown origin) expressed in human HeLa cells transfected with empty vector using [3H]AEA as substrate after 18 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of FAAH (unknown origin) expressed in human HeLa cells using [3H]AEA as substrate after 18 hrsMore data for this Ligand-Target Pair